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Module Name

Medicinal Chemistry Practice

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Code of Subjects

P10A02.0410

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Study load

1(1-0) credits

Contact hour per semester: 13

Total workload : 13

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Semester

4

4

Precondition

P10A.0206

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Competence

After graduating from this course, students are expected to be able to:

1. Able to formulate steps in the development of new drugs
2. Able to practice the steps in the development of new drugs

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Elements of Competency

MKK

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Type Competency

Main competence

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Syllabus

In this course, students learn about practices and technical sequences in the rational discovery and design of new drugs, starting from computational studies and molecular modeling consisting of molecular anchoring, pharmacophore screening, quantitative relationships of structure and activity, preformulation and characterization of the resulting comp

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Attribute Soft Skill

Ethics, awareness, discipline

10

Learning methods

Presentation, lecturer, discussion, project

11

Learning Media

LCD Projector

12

Appraisal

Assignment : 30% 

Mid-Exam : 35%

Final-Exam : 35%

13

Lecturer

Prof. apt. Muchtaridi, M.Si. and Apt. Intan Timur Maesyaroh, Ph.D.

14

References

1. Muchtaridi dkk. 2017, Kimia Medisinal DASAR-DASAR DALAM Perancangan Obat
2. Muchtaridi dkk. 2019, Penambatan Molekul Teori dan Praktek
3. Patrick, G. L. (2017). An Introduction to Medicinal Chemistry. Oxford University Press.
4. Davis, A., & Ward, S. E. (2015). The Handbook of Medicinal Chemistry. In The Handbook of Medicinal Chemistry. Royal Society of Chemistry.
5. Barret, R. (2018). Medicinal Chemistry: Fundamentals. Elsevier Science.
6. Helmer, E. (2016). Textbook of Medicinal Chemistry. Syrawood Publishing House.
7. Wermuth, C. G., Aldous, D., Raboisson, P., & Rognan, D. (2015). The Practice of Medicinal Chemistry. Elsevier Science.
8. Renslo, A. (2016). The organic chemistry of medicinal agents. McGraw-Hill Education.
9. Kumar, T. D. A., & Swathi, N. (2016). Experimental Organic & Medicinal Chemistry: Principles & Practice. Pharma Med Press.
10. Yet, L. (2018). Privileged Structures in Drug Discovery. In Privileged Structures in Drug Discovery. Wiley.
11. Abraham, D. J., & Myers, M. (2021). Burger’s Medicinal Chemistry, Drug Discovery and Development, 8 Volume Set. Wiley.
12. Petitjean, M., & Camproux, A.-C. (2016). In Silico Medicinal Chemistry: Computational Methods to Support Drug Design. Edited by Nathan Brown. In ChemMedChem (Vol. 11, Issue 13). Royal Society of Chemistry.